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Synthesis and Preclinical Evaluation of Sulfonamido-based  [11C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase
Synthesis and Preclinical Evaluation of Sulfonamido-based [11C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase

Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in  cancer malignancy, neurological and metabolic disorders - ScienceDirect
Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in cancer malignancy, neurological and metabolic disorders - ScienceDirect

Potential application of endocannabinoid system agents in neuropsychiatric  and neurodegenerative diseases—focusing on FAAH/MAGL inhibitors | Acta  Pharmacologica Sinica
Potential application of endocannabinoid system agents in neuropsychiatric and neurodegenerative diseases—focusing on FAAH/MAGL inhibitors | Acta Pharmacologica Sinica

Identification of ABX-1431, a Selective Inhibitor of Monoacylglycerol  Lipase and Clinical Candidate for Treatment of Neurological Disorders |  Journal of Medicinal Chemistry
Identification of ABX-1431, a Selective Inhibitor of Monoacylglycerol Lipase and Clinical Candidate for Treatment of Neurological Disorders | Journal of Medicinal Chemistry

Monoacylglycerol lipase (MAGL) as a promising therapeutic target -  ScienceDirect
Monoacylglycerol lipase (MAGL) as a promising therapeutic target - ScienceDirect

Frontiers | Modulation of the Endocannabinoid System as a Potential  Anticancer Strategy
Frontiers | Modulation of the Endocannabinoid System as a Potential Anticancer Strategy

Molecules | Free Full-Text | Targeting Monoacylglycerol Lipase in Pursuit  of Therapies for Neurological and Neurodegenerative Diseases
Molecules | Free Full-Text | Targeting Monoacylglycerol Lipase in Pursuit of Therapies for Neurological and Neurodegenerative Diseases

Chem Soc Rev
Chem Soc Rev

Full article: An updated patent review of monoacylglycerol lipase (MAGL)  inhibitors (2018-present)
Full article: An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)

Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in  cancer malignancy, neurological and metabolic disorders - ScienceDirect
Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in cancer malignancy, neurological and metabolic disorders - ScienceDirect

The highs of endocannabinoid physiology - The Physiological Society
The highs of endocannabinoid physiology - The Physiological Society

A Schematic model of the effects of MAGL inhibition on the interactions...  | Download Scientific Diagram
A Schematic model of the effects of MAGL inhibition on the interactions... | Download Scientific Diagram

Overview of current clinical studies of MAGL inhibitor 21 (ABX-1431). |  Download Scientific Diagram
Overview of current clinical studies of MAGL inhibitor 21 (ABX-1431). | Download Scientific Diagram

Overview of current clinical studies of MAGL inhibitor 21 (ABX-1431). |  Download Scientific Diagram
Overview of current clinical studies of MAGL inhibitor 21 (ABX-1431). | Download Scientific Diagram

Therapeutic endocannabinoid augmentation for mood and anxiety disorders:  comparative profiling of FAAH, MAGL and dual inhibitors | Translational  Psychiatry
Therapeutic endocannabinoid augmentation for mood and anxiety disorders: comparative profiling of FAAH, MAGL and dual inhibitors | Translational Psychiatry

Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in  cancer malignancy, neurological and metabolic disorders - ScienceDirect
Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in cancer malignancy, neurological and metabolic disorders - ScienceDirect

Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective  Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of  Neuroinflammation | Journal of Medicinal Chemistry
Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation | Journal of Medicinal Chemistry

Molecules | Free Full-Text | Discovery of Monoacylglycerol Lipase (MAGL)  Inhibitors Based on a Pharmacophore-Guided Virtual Screening Study
Molecules | Free Full-Text | Discovery of Monoacylglycerol Lipase (MAGL) Inhibitors Based on a Pharmacophore-Guided Virtual Screening Study

Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective  Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of  Neuroinflammation | Journal of Medicinal Chemistry
Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation | Journal of Medicinal Chemistry

Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in  cancer malignancy, neurological and metabolic disorders - ScienceDirect
Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in cancer malignancy, neurological and metabolic disorders - ScienceDirect

Potential application of endocannabinoid system agents in neuropsychiatric  and neurodegenerative diseases—focusing on FAAH/MAGL inhibitors | Acta  Pharmacologica Sinica
Potential application of endocannabinoid system agents in neuropsychiatric and neurodegenerative diseases—focusing on FAAH/MAGL inhibitors | Acta Pharmacologica Sinica

Dual blockade of FAAH and MAGL identifies behavioral processes regulated by  endocannabinoid crosstalk in vivo | PNAS
Dual blockade of FAAH and MAGL identifies behavioral processes regulated by endocannabinoid crosstalk in vivo | PNAS

Molecules | Free Full-Text | Targeting Monoacylglycerol Lipase in Pursuit  of Therapies for Neurological and Neurodegenerative Diseases
Molecules | Free Full-Text | Targeting Monoacylglycerol Lipase in Pursuit of Therapies for Neurological and Neurodegenerative Diseases

Representative small molecule MAGL inhibitors. | Download Scientific Diagram
Representative small molecule MAGL inhibitors. | Download Scientific Diagram

Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in  cancer malignancy, neurological and metabolic disorders
Monoacylglycerol lipase inhibitors: modulators for lipid metabolism in cancer malignancy, neurological and metabolic disorders

Frontiers | Discovering monoacylglycerol lipase inhibitors by a combination  of fluorogenic substrate assay and activity-based protein profiling
Frontiers | Discovering monoacylglycerol lipase inhibitors by a combination of fluorogenic substrate assay and activity-based protein profiling